Paper4613
Dissociation constants and relative efficacies of agonists acting on alpha adrenergic receptors in rabbit aorta.
Besse JC and 1 other. J Pharmacol Exp Ther, 1976. Cited by 257 papers, by iCite.
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ConductScience Library. Dissociation constants and relative efficacies of agonists acting on alpha adrenergic receptors in rabbit aorta. Papers, record 4613. Release papers-2026-11-12-0.1.0, 12 Nov 2026. https://conductscience.org/library/papers/4613
Paper
PubMed's record of the paper, with iCite's citation figures. No abstract is shown.
- Title
- Dissociation constants and relative efficacies of agonists acting on alpha adrenergic receptors in rabbit aorta.
- PubMed
Topics14
NLM's MeSH indexing of the paper, its major topics first.
| MeSH term | Major |
|---|---|
| Adrenergic alpha-Agonists | Major topic |
| Aorta, Thoracic | Major topic |
| Adrenergic beta-Agonists | |
| Animals | |
| Chemical Phenomena | |
| Chemistry | |
| Dibenzylchlorethamine | |
| In Vitro Techniques | |
| Kinetics | |
| Muscle Contraction | |
| Norepinephrine | |
| Phentolamine | |
| Rabbits | |
| Receptors, Adrenergic |
Source PubMed
Cited by38
The papers in our copy of PubMed whose reference list names this one, newest first. iCite, which reads more sources, counts 257 citations.
| PMID | Title | Journal | Year | In Papers | Source |
|---|---|---|---|---|---|
| 32,799,410 | Biochemical characterization of AeD7L2 and its physiological relevance in blood feeding in the dengue mosquito vector, Aedes aegypti. | FEBS J | 2021 | https://conductscience.org/library/papers/32799410 | PubMed |
| 31,412,133 | In vitro determination of the efficacy of illicit synthetic cannabinoids at CB1 receptors. | Br J Pharmacol | 2019 | https://conductscience.org/library/papers/31412133 | PubMed |
| 26,905,519 | Analyzing isolated blood vessel contraction in multi-well plates. | Naunyn Schmiedebergs Arch Pharmacol | 2016 | https://conductscience.org/library/papers/26905519 | PubMed |
| 24,737,484 | A comparison of histamine effects on the sympathetic neurotransmission of testicular capsule and rat vas deferens. | Naunyn Schmiedebergs Arch Pharmacol | 2014 | https://conductscience.org/library/papers/24737484 | PubMed |
| 23,259,038 | Chemical modification of the M(1) agonist VU0364572 reveals molecular switches in pharmacology and a bitopic binding mode. | ACS Chem Neurosci | 2012 | https://conductscience.org/library/papers/23259038 | PubMed |
| 20,590,656 | An operational model of pharmacological agonism: the effect of E/[A] curve shape on agonist dissociation constant estimation. 1985. | Br J Pharmacol | 2010 | https://conductscience.org/library/papers/20590656 | PubMed |
| 19,602,444 | What is the real physiological NO concentration in vivo? | Nitric Oxide | 2009 | https://conductscience.org/library/papers/19602444 | PubMed |
| 18,223,670 | Agonist binding, agonist affinity and agonist efficacy at G protein-coupled receptors. | Br J Pharmacol | 2008 | https://conductscience.org/library/papers/18223670 | PubMed |
| 10,433,496 | Inverse agonist activities of beta-adrenoceptor antagonists in rat myocardium. | Br J Pharmacol | 1999 | https://conductscience.org/library/papers/10433496 | PubMed |
| 8,886,408 | Characterization of alpha 1 D-adrenoceptor subtype in rat myocardium, aorta and other tissues. | Br J Pharmacol | 1996 | https://conductscience.org/library/papers/8886408 | PubMed |
| 8,564,230 | Determination of beta-adrenoceptor subtype on rat isolated ventricular myocytes by use of highly selective beta-antagonists. | Br J Pharmacol | 1995 | https://conductscience.org/library/papers/8564230 | PubMed |
| 8,548,172 | Extended concentration-response curves used to reflect full agonist efficacies and receptor occupancy-response coupling ranges. | Br J Pharmacol | 1995 | https://conductscience.org/library/papers/8548172 | PubMed |
| 7,099,925 | Differences in the development of sensitization to norepinephrine between isolated aortas of untreated and reserpinized rabbits. | Pflugers Arch | 1982 | https://conductscience.org/library/papers/7099925 | PubMed |
| 6,733,356 | Muscarinic receptor occupation and receptor activation in the guinea-pig ileum by some acetamides related to oxotremorine. | Br J Pharmacol | 1984 | https://conductscience.org/library/papers/6733356 | PubMed |
| 6,680,278 | Membrane transport in vascular smooth muscle and its relation to normal and altered excitation during hypertension. | Ann Biomed Eng | 1983 | https://conductscience.org/library/papers/6680278 | PubMed |
| 6,289,955 | Receptor interactions of imidazolines: alpha-adrenoceptors of rat and rabbit aortae differentiated by relative potencies, affinities and efficacies of imidazoline agonists. | Br J Pharmacol | 1982 | https://conductscience.org/library/papers/6289955 | PubMed |
| 6,289,140 | Analysis of the beta 1 and beta 2 adrenoceptor interactions of the partial agonist, clenbuterol (NAB365), in the rat jugular vein and atria. | Naunyn Schmiedebergs Arch Pharmacol | 1982 | https://conductscience.org/library/papers/6289140 | PubMed |
| 6,140,043 | Temperature-induced changes in dissociation constants (KA) of agonists at cardiac beta-adrenoceptors determined by use of the irreversible antagonist Ro 03-7894. | Br J Pharmacol | 1983 | https://conductscience.org/library/papers/6140043 | PubMed |
| 6,116,509 | Dissociation constants of isoprenaline and orciprenaline and their relative efficacies on guinea-pig isolated atria determined by use of an irreversible beta-adrenoceptor antagonist. | Br J Pharmacol | 1981 | https://conductscience.org/library/papers/6116509 | PubMed |
| 3,978,322 | An operational model of pharmacological agonism: the effect of E/[A] curve shape on agonist dissociation constant estimation. | Br J Pharmacol | 1985 | https://conductscience.org/library/papers/3978322 | PubMed |
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- 2026-11-12
- Gene search
- 2026-11-11
- Pipelines
- 2026-09-18
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- ChEMBL, through Open TargetsCC BY-SA 3.0
- ClinicalTrials.govNo license stated
- HGNCCC0
- iCiteCC BY 4.0
- NCBI GenePublic domain (US government)
- NIH RePORTER's grant and paper linksPublic domain
- Open TargetsCC0 1.0
- PMC's ID filePublic domain (US government)
- PubMedNLM's terms
- PubTator 3Public domain
- UniProtCC BY 4.0
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- ChEMBL, through Open TargetsCC BY-SA 3.0, for the parts from ChEMBL. Read on 8 Nov 2026 at https://platform-docs.opentargets.org/licence
- ClinicalTrials.govnone stated
- HGNCCC0: https://www.genenames.org/about/license/
- iCiteCC BY 4.0
- NCBI GeneNone named for the file. NCBI says information created by or for the US government on its site is in the public domain, and asks that NLM be acknowledged: https://www.ncbi.nlm.nih.gov/home/about/policies/
- NIH RePORTER's grant and paper linksPublic domain (NIH RePORTER)
- Open TargetsCC0 1.0. Open Targets asks that users cite its latest paper: Buniello et al. 2025, Open Targets Platform: facilitating therapeutic hypotheses building in drug discovery, Nucleic Acids Research 53(D1):D1467, PMID 39657122. Read on 8 Nov 2026 at https://platform-docs.opentargets.org/licence
- PMC's ID fileNone named for the file. NCBI says information created by or for the US government on its site is in the public domain, and asks that NLM be acknowledged: https://www.ncbi.nlm.nih.gov/home/about/policies/
- PubMedNLM's terms
- PubTator 3Public domain
- UniProtCC BY 4.0. UniProt's licence file: "All databases and documents in the UniProt FTP directory may be copied and redistributed freely, without advance permission, provided that this copyright statement is reproduced with each copy." UniProt asks that users cite its latest paper: The UniProt Consortium, UniProt: the Universal Protein Knowledgebase in 2025, Nucleic Acids Research 53:D609-D617, https://doi.org/10.1093/nar/gkae1010. Read on 9 Nov 2026 at https://www.uniprot.org/help/license
ClinicalTrials.gov's data carry an international copyright outside the United States: https://clinicaltrials.gov/about-site/terms-conditions.
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